SCHEMBL5223628

SCHEMBL5223628

CC(=O)c1c(C)[nH]c(C(=O)O)c1C#N

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
MAPT P10636 3/20 0.43
GAA P10253 2/20 0.43
CREBBP Q92793 3/20 0.42
BRD4 O60885 2/20 0.42
BRPF1 P55201 2/20 0.42
ESR1 P03372 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPSR1 Q6W5P4 2/20 0.39
EP300 Q09472 1/20 0.38
KMT2A Q03164 2/20 0.38
HPGD P15428 2/20 0.37
MEN1 O00255 1/20 0.37
HSD17B10 Q99714 1/20 0.37
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPK1 P28482 3/20 0.37
SMN1; SMN2 Q16637 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5279994 0.84 CYP1A2 (0.47) CYP1A2CYP3A4MAPTGAACREBBP
SCHEMBL510531 0.76 KDM4E (0.49) CYP3A4MAPTGAAKMT2AHPGD
SCHEMBL399174 0.76 ATM (0.49) MAPTGAANPSR1KMT2AHPGD
SCHEMBL3033303 0.76 ALDH1A1 (0.40) CYP1A2CYP3A4MAPTGAAESR1
SCHEMBL1411774 0.75 CYP1A2 (0.76) CYP1A2CYP3A4MAPTCREBBPBRD4
SCHEMBL3399851 0.73 KDM4E (0.44) CYP3A4MAPTGAANPSR1KMT2A
SCHEMBL401727 0.73 ATM (0.44) MAPTGAANPSR1KMT2AHPGD
SCHEMBL10815675 0.71 KDM4E (0.56) CYP1A2CYP3A4MAPTGAACREBBP
SCHEMBL2150911 0.71 CYP1A2 (0.57) CYP1A2CYP3A4MAPTCREBBPBRD4
SCHEMBL11018436 0.70 KDM4E (0.46) CYP1A2CYP3A4MAPTGAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664025-B1 PYRROL DERIVATIVES WITH ANTIBACTERIAL ACTIVITY ASTRAZENECA AB (SE) 2007-09-19 EP disclosed
EP-1363925-B1 MACROLIDE ANTIBIOTICS GLAXO GROUP LTD (GB) 2006-11-15 EP disclosed