SCHEMBL5223852

SCHEMBL5223852

O=c1c2ncc3c(c(CNCCc4ccccc4)cn3Cc3ccc(F)cc3)c2ccn1O

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 3/20 0.41
KMT2A Q03164 3/20 0.39
HASPIN Q8TF76 1/20 0.39
SLC6A5 Q9Y345 1/20 0.38
TRPV6 Q9H1D0 1/20 0.37
FYN P06241 1/20 0.37
SRC P12931 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TSHR P16473 1/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
TP53 P04637 1/20 0.36
PLA2G4A P47712 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
DRD2 P14416 1/20 0.36
HTR6 P50406 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14302890 0.90 KDM4E (0.43) ALDH1A1KDM4EKMT2ASMN1; SMN2LMNA
SCHEMBL3495823 0.89 MCHR1 (0.36) ALDH1A1KDM4EKMT2ASMN1; SMN2TP53
SCHEMBL14303283 0.88 KDM4E (0.36) ALDH1A1KDM4EKMT2ASMN1; SMN2
SCHEMBL3495444 0.85 TP53 (0.41) ALDH1A1KDM4EKMT2ASMN1; SMN2LMNA
SCHEMBL4965499 0.85 KDM4E (0.33) ALDH1A1KDM4EKMT2ASMN1; SMN2
SCHEMBL14395082 0.85 MDM4 (0.34) ALDH1A1KDM4EKMT2ASMN1; SMN2TSHR
SCHEMBL14302885 0.85 ALDH1A1 (0.37) ALDH1A1KDM4EKMT2ASMN1; SMN2TP53
SCHEMBL4962801 0.84 KDM4E (0.34) ALDH1A1KDM4EKMT2ASMN1; SMN2CNR2
SCHEMBL3495927 0.84 POLB (0.42) KDM4EKMT2ALMNAHPGDTP53
SCHEMBL4964868 0.83 CYP19A1 (0.39) ALDH1A1KDM4EKMT2ASMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751157-B1 INHIBITORS OF THE HIV INTEGRASE ENZYME PFIZER (US) 2007-10-03 EP claimed