SCHEMBL5223929

SCHEMBL5223929

COc1ccc(C(=O)Nc2ccccc2NC(=O)c2ccc(OC)cc2OCc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.68
KDM4E B2RXH2 3/20 0.68
CYP1A2 P05177 1/20 0.68
CYP2C9 P11712 1/20 0.68
CYP2C19 P33261 1/20 0.68
F10 P00742 2/20 0.61
PPARD Q03181 1/20 0.60
NPC1 O15118 6/20 0.56
RAB9A P51151 6/20 0.56
SMN1; SMN2 Q16637 3/20 0.56
GAA P10253 1/20 0.56
CASP3 P42574 2/20 0.56
SENP7 Q9BQF6 2/20 0.56
TAAR1 Q96RJ0 1/20 0.56
MAPT P10636 2/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
ABCG2 Q9UNQ0 1/20 0.54
LMNA P02545 1/20 0.54
HTT P42858 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1123360 0.82 KDM4E (0.62) ALDH1A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL2295551 0.80 NPC1 (0.71) ALDH1A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL7251634 0.79 KDM4E (0.54) ALDH1A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL38660966 0.79 MEN1 (0.60) ALDH1A1KDM4ECYP1A2CYP2C9CYP2C19
SCHEMBL11557673 0.79 KDM4E (0.60) KDM4ENPC1RAB9ASMN1; SMN2GAA
SCHEMBL31550547 0.79 HDAC8 (0.60) KDM4ENPC1RAB9ASMN1; SMN2GAA
SCHEMBL6404086 0.79 HDAC8 (0.60) KDM4ENPC1RAB9ASMN1; SMN2GAA
SCHEMBL3821744 0.78 F10 (0.93) ALDH1A1F10NPC1RAB9ASMN1; SMN2
SCHEMBL28249518 0.78 POLB (0.67) ALDH1A1KDM4ECYP1A2CYP2C19NPC1
SCHEMBL6450099 0.78 MAOB (0.65) ALDH1A1KDM4ECYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1014962-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2007-06-27 EP disclosed
EP-1014962-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-07-05 EP disclosed
WO-1999000121-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1999-01-07 WO disclosed