SCHEMBL5224314

SCHEMBL5224314

COC(=O)[C@@H]1CSCN1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3361966 1.00
SCHEMBL11122946 1.00
Hydrochloric Acid SCHEMBL201249 0.98 KMT2A (0.41)
Hydrochloric Acid SCHEMBL201248 0.98 KMT2A (0.41)
Hydrochloric Acid SCHEMBL7350919 0.98 KMT2A (0.41)
Hydrochloric Acid SCHEMBL6392619 0.96 KMT2A (0.40)
Hydrochloric Acid SCHEMBL6395633 0.96 KMT2A (0.40)
SCHEMBL28052844 0.83
SCHEMBL4571091 0.82 KMT2A (0.41)
SCHEMBL5493487 0.82 KMT2A (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024044098-A2 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS ALEXION PHARMACEUTICALS, INC. (US) 2024-02-29 WO disclosed
US-20230348493-A1 COMPOUND FOR ADJUSTING ACTIVITY OF NMDA RECEPTOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF BEIJING GREATWAY PHARMACEUTICAL TECHNOLOGY CO. LTD. (CN) 2023-11-02 US disclosed
CN-104447947-A Process for producing pidotimod CHENGDU YILUKANG MEDICAL TECHNOLOGY & SERVICE CO L 2015-03-25 CN disclosed
EP-1406872-B1 DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OF DIABETES MERCK & CO INC (US) 2007-12-19 EP disclosed
US-7098239-B2 Dipeptidyl peptidase inhibitors for the treatment of diabetes MERCK & CO., INC (US) 2006-08-29 US disclosed
EP-1406872-A4 DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OF DIABETES MERCK & CO INC (US) 2005-01-19 EP disclosed
US-20040176428-A1 Dipeptidyl peptidase inhibitors for the treatment of diabetes MERCK SHARP & DOHME CORP. 2004-09-09 US disclosed
EP-1406872-A2 DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OF DIABETES Merck & Co., Inc. (US) 2004-04-14 EP disclosed
WO-2003000180-A2 DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OF DIABETES MERCK & CO., INC. (US) 2003-01-03 WO disclosed
EP-0461677-B1 Novel thiazolidine derivatives ONO PHARMACEUTICAL CO (JP) 1997-04-16 EP disclosed
EP-0280956-B1 THIAZOLIDINE DERIVATIVES ONO PHARMACEUTICAL CO., LTD. (JP) 1992-10-21 EP disclosed
CN-1017435-B PROCESS FOR PREPARATION OF GLYCEROL DERIVATIVES NIPPON CHEMIPHAR CO (JP) 1992-07-15 CN disclosed
EP-0461677-A1 Novel thiazolidine derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 1991-12-18 EP disclosed
US-4857537-A PREVENTING AMNESIA ONO PHARMACEUTICAL CO., LTD. (JP) 1989-08-15 US disclosed
CN-1030239-A The preparation method of new glycerol derivative NIPPON CHEMIPHAR CO (JP) 1989-01-11 CN disclosed
EP-0280956-A1 Thiazolidine derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 1988-09-07 EP disclosed