SCHEMBL5225318

SCHEMBL5225318

Cc1ccc(Nc2nccc(CNc3ccc4c(c3)nc(NC(=O)Cc3ccc(Cl)c(Cl)c3)n4C)n2)cc1S(N)(=O)=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 2/20 0.43
HTT P42858 1/20 0.43
BTK Q06187 1/20 0.41
MTOR P42345 1/20 0.39
KDR P35968 4/20 0.37
AURKB Q96GD4 3/20 0.37
CYP3A4 P08684 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP2C9 P11712 2/20 0.37
CYP2C19 P33261 2/20 0.37
PTK2 Q05397 2/20 0.37
PLK4 O00444 2/20 0.37
AURKA O14965 2/20 0.37
JAK2 O60674 2/20 0.37
MAP4K4 O95819 2/20 0.37
LCK P06239 2/20 0.37
FYN P06241 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5223137 0.85 KDR (0.56) SMN1; SMN2ALDH1A1LMNAMAPTHTT
SCHEMBL4978591 0.78 KDR (0.45) SMN1; SMN2ALDH1A1LMNAMAPTHTT
SCHEMBL4978600 0.74 LMNA (0.46) SMN1; SMN2ALDH1A1LMNAMAPTHTT
SCHEMBL4978336 0.73 KDR (0.45) KDRMET
SCHEMBL4977088 0.73 KDR (0.40) KDRMETNTRK1
SCHEMBL4980837 0.73 BTK (0.50) SMN1; SMN2BTKMTORKDRAURKB
SCHEMBL5224590 0.72 KDR (0.54) KDRAURKBCYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL4980031 0.72 BTK (0.49) SMN1; SMN2BTKMTORKDRAURKB
SCHEMBL5225921 0.72 KDR (0.55) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5225412 0.71 KDR (0.55) KDRAURKBCYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP disclosed