SCHEMBL5225564

SCHEMBL5225564

CN(c1ccc2c(c1)nc(-c1ccccc1N(C(=O)O)C(C)(C)C)n2C)c1ccnc(Cl)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.38
CYP3A4 P08684 2/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
HPGD P15428 1/20 0.35
KIT P10721 6/20 0.33
PDGFRA P16234 5/20 0.33
AGPAT2 O15120 2/20 0.33
HDAC1 Q13547 5/20 0.32
HDAC8 Q9BY41 5/20 0.32
HDAC6 Q9UBN7 5/20 0.32
HDAC3 O15379 4/20 0.32
HDAC4 P56524 4/20 0.32
HDAC7 Q8WUI4 4/20 0.32
HDAC2 Q92769 4/20 0.32
HDAC10 Q969S8 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226754 0.84 KDR (0.39) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5222711 0.82 KDR (0.42) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5225347 0.81 KDR (0.37) KDRCYP2C9KDM4EALDH1A1CYP1A2
SCHEMBL5225821 0.81 KDR (0.57) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5227034 0.80 KDR (0.68) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5225575 0.78 KDR (0.36) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5222688 0.77 KDR (0.40) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5227351 0.76 KDR (0.44) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5225570 0.76 KDR (0.41) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5228803 0.75 KDR (0.40) KDRCYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP disclosed