SCHEMBL5225347

SCHEMBL5225347

Cn1c(-c2ccccc2N(C(=O)O)C(C)(C)C)nc2cc(Nc3ccnc(Cl)n3)ccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.37
PTK2 Q05397 2/20 0.37
PLK1 P53350 1/20 0.37
AURKB Q96GD4 1/20 0.37
AGPAT2 O15120 3/20 0.37
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
P2RX3 P56373 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
HPGD P15428 1/20 0.35
AKT1 P31749 1/20 0.35
BRAF P15056 3/20 0.34
NAMPT P43490 1/20 0.34
CYP2C9 P11712 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225564 0.81 KDR (0.38) KDRAGPAT2KDM4EALDH1A1CYP1A2
SCHEMBL5225363 0.79 RAF1 (0.39) KDRAURKBNPC1RAB9APOLB
SCHEMBL5227201 0.76 BRAF (0.48) KDRNPC1RAB9APOLBMAPT
SCHEMBL5225357 0.75 NPC1 (0.40) KDRPTK2PLK1AURKBAGPAT2
SCHEMBL5223899 0.74 ALDH1A1 (0.45) NPC1RAB9AMAPTKDM4EALDH1A1
SCHEMBL4980380 0.73 BRAF (0.37) KDRAURKBNPC1RAB9APOLB
SCHEMBL5228478 0.73 NPC1 (0.41) AGPAT2NPC1RAB9APOLBMAPT
SCHEMBL5226236 0.73 BRAF (0.45) KDRNPC1RAB9APOLBMAPT
SCHEMBL588578 0.73 RAB9A (0.52) NPC1RAB9APOLBMAPTKDM4E
SCHEMBL5227034 0.71 KDR (0.68) KDRPTK2AURKBCYP1A2BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP disclosed