SCHEMBL5225717

SCHEMBL5225717

CC(=Cc1ccc(N)c(N)c1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.55
SLC9A1 P19634 1/20 0.40
SLC9A3 P48764 1/20 0.40
SLC9A2 Q9UBY0 1/20 0.40
TBXAS1 P24557 6/20 0.39
APEX1 P27695 7/20 0.36
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35
TUBA4A P68366 1/20 0.35
TUBB4B P68371 1/20 0.35
TUBB3 Q13509 1/20 0.35
TUBB2A Q13885 1/20 0.35
TUBB8 Q3ZCM7 1/20 0.35
TUBA3E Q6PEY2 1/20 0.35
TUBA1A Q71U36 1/20 0.35
TUBA1C Q9BQE3 1/20 0.35
TUBB6 Q9BUF5 1/20 0.35
TUBB2B Q9BVA1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225714 1.00 AKR1C3 (0.55) AKR1C3SLC9A1SLC9A3SLC9A2TBXAS1
SCHEMBL14086414 0.86 AKR1C3 (0.52) AKR1C3SLC9A1SLC9A3SLC9A2TBXAS1
SCHEMBL15709486 0.82 AKR1C3 (0.47) AKR1C3SLC9A1SLC9A3SLC9A2TBXAS1
SCHEMBL10634979 0.82 APP (0.51) AKR1C3APEX1TUBB4ATUBBTUBA3C
SCHEMBL15709484 0.82 AKR1C3 (0.47) AKR1C3SLC9A1SLC9A3SLC9A2TBXAS1
SCHEMBL10634987 0.82 APP (0.51) AKR1C3APEX1TUBB4ATUBBTUBA3C
SCHEMBL2462983 0.80 AKR1C3 (0.82) AKR1C3TBXAS1APEX1KDM4EGLA
SCHEMBL2462984 0.80 AKR1C3 (0.82) AKR1C3TBXAS1APEX1KDM4EGLA
SCHEMBL8746638 0.79 AKR1C3 (0.61) AKR1C3SLC9A1SLC9A3SLC9A2TBXAS1
SCHEMBL3033605 0.79 AKR1C3 (0.67) AKR1C3TBXAS1APEX1KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758857-A1 INDOLE DERIVATIVES AS ANTIVIRAL AGENTS Istituto di Richerche di Biologia Molecolare P. Angeletti S.p.A. (IT) 2007-03-07 EP disclosed
WO-2006029912-A1 INDOLE DERIVATIVES AS ANTIVIRAL AGENTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI SPA (IT) 2006-03-23 WO disclosed