SCHEMBL5225728

SCHEMBL5225728

CN1CCN(CCCNC(=O)Oc2nc(-c3ccc(S(=O)(=O)N4CCCC4)cc3)cnc2N)CC1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 17/20 0.60
CCNE2 O96020 12/20 0.60
CCNE1 P24864 12/20 0.60
CDK2 P24941 12/20 0.60
GSK3A P49840 1/20 0.47
ALDH1A1 P00352 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.42
RECQL P46063 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ROCK2 O75116 1/20 0.42
ROCK1 Q13464 1/20 0.42
KCNH2 Q12809 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5219446 0.91 GSK3B (0.51) GSK3BCCNE2CCNE1CDK2ALDH1A1
Hydrochloric Acid SCHEMBL5221093 0.87 GSK3B (0.77) GSK3BCCNE2CCNE1CDK2GSK3A
Hydrochloric Acid SCHEMBL5219189 0.86 GSK3B (0.58) GSK3BCCNE2CCNE1CDK2GSK3A
Hydrochloric Acid SCHEMBL5224554 0.86 GSK3B (0.61) GSK3BCCNE2CCNE1CDK2GSK3A
Hydrochloric Acid SCHEMBL5223613 0.86 GSK3B (0.61) GSK3BCCNE2CCNE1CDK2GSK3A
SCHEMBL3274547 0.86 GSK3B (0.78) GSK3BCCNE2CCNE1CDK2GSK3A
Hydrochloric Acid SCHEMBL5224249 0.85 GSK3B (0.49) GSK3BCCNE2CCNE1CDK2ALDH1A1
Hydrochloric Acid SCHEMBL5223643 0.85 GSK3B (0.61) GSK3BCCNE2CCNE1CDK2GSK3A
SCHEMBL5221380 0.85 GSK3B (0.51) GSK3BCCNE2CCNE1CDK2GSK3A
Hydrochloric Acid SCHEMBL5223876 0.84 CYP1A2 (0.58) GSK3BCCNE2CCNE1CDK2GSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575942-B1 COMPOUNDS HAVING SELECTIVE INHIBITING EFECT AT GSK3 ASTRAZENECA AB (SE) 2007-05-02 EP claimed