SCHEMBL5225849

SCHEMBL5225849

Cc1ccc(Nc2nccc(N(C)c3ccc4c(c3)nc(-c3c(NC(=O)O)cccc3C(C)(C)C)n4C)n2)cc1S(N)(=O)=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 17/20 0.57
CYP3A4 P08684 8/20 0.57
CYP2D6 P10635 8/20 0.57
CYP2C9 P11712 8/20 0.57
CYP2C19 P33261 8/20 0.57
RIPK1 Q13546 3/20 0.57
RIPK3 Q9Y572 3/20 0.57
KIT P10721 3/20 0.57
CSF1R P07333 3/20 0.57
FLT1 P17948 3/20 0.57
FLT4 P35916 3/20 0.57
ABCB11 O95342 2/20 0.57
PDGFRB P09619 2/20 0.57
FGFR1 P11362 2/20 0.57
AURKA O14965 2/20 0.57
PDGFRA P16234 2/20 0.57
STK16 O75716 2/20 0.57
MAP3K11 Q16584 2/20 0.57
TAOK2 Q9UL54 2/20 0.57
BMPR1B O00238 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227042 0.92 KDR (0.69) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL5228442 0.88 KDR (0.59) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5225853 0.84 KDR (0.56) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5225570 0.82 KDR (0.41) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL14419332 0.81 KDR (0.77) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL5226467 0.81 KDR (0.60) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5225821 0.81 KDR (0.57) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4981197 0.80 KDR (0.69) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL5226899 0.80 KDR (0.72) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4977022 0.80 KDR (0.64) KDRCYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP claimed