SCHEMBL5227042

SCHEMBL5227042

CN(c1ccc2c(c1)nc(-c1c(NC(=O)O)cccc1C(C)(C)C)n2C)c1ccnc(Nc2cccc(S(N)(=O)=O)c2)n1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 18/20 0.69
CYP3A4 P08684 8/20 0.69
CYP2D6 P10635 8/20 0.69
CYP2C9 P11712 8/20 0.69
CYP2C19 P33261 8/20 0.69
RIPK1 Q13546 3/20 0.52
RIPK3 Q9Y572 3/20 0.52
MLKL Q8NB16 2/20 0.52
AURKA O14965 2/20 0.52
KIT P10721 6/20 0.46
PDGFRA P16234 5/20 0.46
CSF1R P07333 2/20 0.46
PDGFRB P09619 2/20 0.46
FGFR1 P11362 2/20 0.46
FLT1 P17948 2/20 0.46
FLT4 P35916 2/20 0.46
BMPR1B O00238 1/20 0.46
PLK4 O00444 1/20 0.46
GAK O14976 1/20 0.46
EPHB6 O15197 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225849 0.92 KDR (0.57) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL5226899 0.88 KDR (0.72) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5227046 0.84 KDR (0.66) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL588536 0.82 KDR (1.00) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5227034 0.82 KDR (0.68) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5225570 0.82 KDR (0.41) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4980358 0.81 KDR (0.81) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Trifluoroacetic Acid SCHEMBL4982202 0.80 KDR (0.72) KDRCYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL5226870 0.80 KDR (0.72) KDRCYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL4978608 0.80 KDR (0.82) KDRCYP3A4CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487824-B1 DIAMINO-PYRIMIDINES AND THEIR USE AS ANGIOGENESIS INHIBITORS SMITHKLINE BEECHAM CORP (US) 2007-06-20 EP claimed