SCHEMBL5226032

SCHEMBL5226032

CN1CCN(Cc2cnn(-c3ccc(-c4cc(F)ccc4F)cc3)c2-c2ccco2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 3/20 0.39
S1PR1 P21453 2/20 0.38
TNIK Q9UKE5 1/20 0.37
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
MET P08581 1/20 0.36
CHKA P35790 2/20 0.36
MPO P05164 1/20 0.35
SSTR5 P35346 1/20 0.35
CXCR3 P49682 1/20 0.35
DRD4 P21917 3/20 0.35
DRD3 P35462 3/20 0.35
DRD2 P14416 2/20 0.35
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34
JAK3 P52333 1/20 0.34
MAPK14 Q16539 1/20 0.34
PTGS1 P23219 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228457 0.90 PIK3R1 (0.39) SMOALDH1A1METCHKASSTR5
SCHEMBL2761009 0.90 SMO (0.43) SMOTNIKALDH1A1LMNAMET
SCHEMBL5744201 0.89 CHKA (0.41) SMOTNIKALDH1A1LMNAGAA
SCHEMBL5224673 0.87 SMO (0.40) SMOTNIKALDH1A1LMNAMET
SCHEMBL2001547 0.87 SMO (0.40) SMOTNIKALDH1A1LMNAGAA
SCHEMBL7261026 0.86 SMO (0.41) SMOS1PR1TNIKALDH1A1CHKA
SCHEMBL2000028 0.86 USP7 (0.39) SMOTNIKALDH1A1LMNAGAA
SCHEMBL1995720 0.85 SMO (0.38) SMOTNIKALDH1A1LMNAGAA
SCHEMBL12569255 0.82 SMO (0.39) SMOALDH1A1LMNAGAASSTR5
SCHEMBL5224366 0.82 SMO (0.44) SMOS1PR1ALDH1A1LMNADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed