SCHEMBL5224673

SCHEMBL5224673

CN1CCN(Cc2cnn(-c3ccc(-c4cccc(F)c4)cc3)c2-c2ccco2)CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 3/20 0.40
KDM1A O60341 1/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
MET P08581 1/20 0.37
ALPL P05186 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 1/20 0.36
DHODH Q02127 1/20 0.36
DRD4 P21917 3/20 0.35
DRD3 P35462 3/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
TYK2 P29597 1/20 0.35
JAK3 P52333 1/20 0.35
DRD2 P14416 2/20 0.35
MAPK14 Q16539 1/20 0.35
PIK3R1 P27986 1/20 0.35
PIK3CA P42336 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5226613 0.93 SMO (0.40) SMOALPLKDM4EALDH1A1LMNA
SCHEMBL2761009 0.91 SMO (0.43) SMOMETALDH1A1LMNADRD4
SCHEMBL5224744 0.89 HTR1A (0.38) SMOALPLKDM4EALDH1A1LMNA
SCHEMBL5226032 0.87 SMO (0.39) SMOMETALDH1A1LMNADRD4
SCHEMBL5229287 0.87 EGFR (0.40) SMOMETALPLKDM4EALDH1A1
SCHEMBL5226986 0.87 DRD4 (0.39) SMOALPLKDM4EALDH1A1LMNA
SCHEMBL5222920 0.85 ALDH1A1 (0.41) KDM4EALDH1A1LMNA
SCHEMBL5230509 0.84 POLB (0.41) SMOMETKDM4EALDH1A1DRD4
SCHEMBL5228457 0.84 PIK3R1 (0.39) SMOKDM1AMAOAMAOBMET
SCHEMBL5228047 0.84 HTR2C (0.37) ALPLKDM4EALDH1A1DHODHDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed