SCHEMBL5228044

SCHEMBL5228044

CC(C)(C)OC(=O)N1CCn2nc(C(F)(F)F)nc2C1COCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.39
DPP4 P27487 7/20 0.39
DPP7 Q9UHL4 6/20 0.39
DPP8 Q6V1X1 3/20 0.39
DPP9 Q86TI2 3/20 0.39
PARP1 P09874 1/20 0.39
KLK7 P49862 1/20 0.37
PDK1 Q15118 1/20 0.36
PDK2 Q15119 1/20 0.36
PDK3 Q15120 1/20 0.36
PDK4 Q16654 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NR1H2 P55055 2/20 0.35
NR1H3 Q13133 2/20 0.35
GAA P10253 1/20 0.35
THRB P10828 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227191 0.87 PARP1 (0.39) DPP4DPP7DPP8DPP9PARP1
SCHEMBL5228676 0.81 DPP4 (0.41) TACR1DPP4DPP7DPP8DPP9
SCHEMBL5227629 0.80 DPP4 (0.37) DPP4DPP7DPP8DPP9NR1H2
SCHEMBL5228855 0.75 DPP4 (0.49) DPP4DPP7DPP8DPP9
SCHEMBL29229139 0.73 KLK7 (0.46) DPP4PARP1KLK7MEN1KMT2A
SCHEMBL29229186 0.73 KLK7 (0.46) DPP4PARP1KLK7MEN1KMT2A
SCHEMBL28549464 0.72 PARP1 (0.46) PARP1KLK7NR1H2NR1H3JAK2
SCHEMBL7921498 0.71 KLK7 (0.47) PARP1KLK7NR1H2NR1H3JAK2
SCHEMBL7921496 0.71 KLK7 (0.47) PARP1KLK7NR1H2NR1H3JAK2
SCHEMBL1341573 0.70 PARP1 (0.40) TACR1PARP1KLK7NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554280-B1 ANTIDIABETIC BETA-AMINO HETEROCYCLIC DIPEPTIDYL PEPTIDASE INHIBITORS MERCK & CO INC (US) 2007-08-15 EP disclosed