SCHEMBL5227191

SCHEMBL5227191

CC(C)(C)OC(=O)N1CCn2nc(C(F)(F)F)nc2C1CC(=O)OCc1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.39
PDK1 Q15118 1/20 0.39
PDK2 Q15119 1/20 0.39
PDK3 Q15120 1/20 0.39
PDK4 Q16654 1/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
DPP4 P27487 6/20 0.38
DPP7 Q9UHL4 6/20 0.38
DPP8 Q6V1X1 3/20 0.38
DPP9 Q86TI2 3/20 0.38
KLK7 P49862 1/20 0.36
HTT P42858 1/20 0.36
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5228044 0.87 TACR1 (0.39) PARP1PDK1PDK2PDK3PDK4
SCHEMBL5228754 0.76 GLA (0.51) PDK1PDK2PDK3PDK4KMT2A
SCHEMBL5228855 0.74 DPP4 (0.49) DPP4DPP7DPP8DPP9ALDH1A1
SCHEMBL344679 0.73 ABCB1 (0.48) PARP1PDK1PDK2PDK3PDK4
SCHEMBL344678 0.73 ABCB1 (0.48) PARP1PDK1PDK2PDK3PDK4
SCHEMBL9037209 0.70 KLK7 (0.51) PARP1KMT2AMEN1KLK7HTT
SCHEMBL24109207 0.69 ABCB1 (0.44) PARP1PDK1PDK2PDK3PDK4
SCHEMBL30315793 0.69 PDK1 (0.51) PARP1PDK1PDK2PDK3PDK4
SCHEMBL30315726 0.69 PDK1 (0.51) PARP1PDK1PDK2PDK3PDK4
SCHEMBL5233907 0.68 DPP4 (0.54) DPP4DPP7DPP8DPP9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1554280-B1 ANTIDIABETIC BETA-AMINO HETEROCYCLIC DIPEPTIDYL PEPTIDASE INHIBITORS MERCK & CO INC (US) 2007-08-15 EP disclosed