SCHEMBL5228832

SCHEMBL5228832

O=C(O)Oc1sc2cc(F)ccc2c1Cl

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCKDK O14874 2/20 0.61
KDM4E B2RXH2 1/20 0.50
LMNA P02545 3/20 0.48
ALDH1A1 P00352 1/20 0.48
RECQL P46063 1/20 0.48
RAB9A P51151 4/20 0.48
SENP1 Q9P0U3 1/20 0.45
TLR3 O15455 1/20 0.44
SMN1; SMN2 Q16637 3/20 0.43
NPC1 O15118 2/20 0.43
TSHR P16473 2/20 0.43
TP53 P04637 1/20 0.43
MCL1 Q07820 2/20 0.43
BCL2L1 Q07817 1/20 0.43
PTGS1 P23219 1/20 0.43
MAOB P27338 1/20 0.43
CASP3 P42574 1/20 0.43
GPER1 Q99527 1/20 0.43
RXFP1 Q9HBX9 2/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16862081 0.87 BCKDK (0.56) BCKDKKDM4ELMNAALDH1A1RECQL
SCHEMBL19283514 0.84 MCL1 (0.59) BCKDKKDM4ELMNAALDH1A1RAB9A
SCHEMBL5237770 0.78 MCL1 (0.57) KDM4ELMNAALDH1A1RAB9ASMN1; SMN2
SCHEMBL5234250 0.77 MAPT (0.56) BCKDKKDM4ELMNAALDH1A1RAB9A
SCHEMBL594468 0.76 BCKDK (1.00) BCKDKKDM4ELMNAALDH1A1RECQL
SCHEMBL2610278 0.75 BCKDK (0.74) BCKDKKDM4ELMNAALDH1A1RECQL
SCHEMBL693146 0.75 BCKDK (0.68) BCKDKKDM4ELMNAALDH1A1RECQL
SCHEMBL2279755 0.73 BCKDK (0.77) BCKDKKDM4ELMNAALDH1A1RECQL
SCHEMBL9203348 0.73 MCL1 (0.57) BCKDKKDM4ELMNAALDH1A1RAB9A
SCHEMBL18187797 0.73 BCKDK (0.61) BCKDKKDM4ELMNAALDH1A1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461335-B1 2-HETEROARYLCARBOXYLIC ACID AMIDES BAYER HEALTHCARE AG (DE) 2007-02-28 EP disclosed
EP-1461335-A1 2-HETEROARYLCARBOXYLIC ACID AMIDES Bayer HealthCare AG (DE) 2004-09-29 EP disclosed
WO-2003055878-A1 2-HETEROARYLCARBOXYLIC ACID AMIDES BAYER HEALTHCARE AG (DE) 2003-07-10 WO disclosed