SCHEMBL5229148

SCHEMBL5229148

CC(Cc1cccc(CC(C)(C)C)c1)NC[C@H](O)[C@H](Cc1cc(F)cc(F)c1)NC(=O)CF

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 20/20 0.54
CTSD P07339 15/20 0.54
BACE2 Q9Y5Z0 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5713938 0.83 CTSD (0.67) BACE1CTSD
SCHEMBL3177017 0.83 CTSD (0.67) BACE1CTSD
SCHEMBL3167952 0.83 CTSD (0.67) BACE1CTSD
SCHEMBL4262818 0.80 BACE1 (0.52) BACE1CTSDBACE2
SCHEMBL3172063 0.76 BACE1 (0.80) BACE1CTSD
SCHEMBL3172074 0.76 BACE1 (0.80) BACE1CTSD
SCHEMBL3502935 0.76 BACE1 (0.80) BACE1CTSD
SCHEMBL13315982 0.76 BACE1 (0.68) BACE1CTSD
Hydrochloric Acid SCHEMBL3172335 0.75 BACE1 (0.67) BACE1CTSD
Hydrochloric Acid SCHEMBL3172343 0.75 BACE1 (0.67) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565443-A4 ACETYL 2-HYDROXY-1,3 DIAMINOALKANES ELAN PHARM INC (US) 2007-07-18 EP claimed
JP-2006504793-A 2006-02-09 JP claimed
EP-1565443-A2 ACETYL 2-HYDROXY-1,3 DIAMINOALKANES Elan Pharmaceuticals, Inc. (US) 2005-08-24 EP claimed
WO-2004024081-A2 ACETYL 2-HYDROXY-1,3 DIAMINOALKANES ELAN PHARMACEUTICALS, INC. (US) 2004-03-25 WO claimed