SCHEMBL5229660

SCHEMBL5229660

Cc1nc(/C=C(/F)[C@@H](O)CC(=O)N2C(=O)O[C@H](c3ccccc3)[C@@H]2C)cs1

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 2/20 0.31
PTGDR2 Q9Y5Y4 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227605 0.89 IDH1 (0.31) IDH1
SCHEMBL5227610 0.89 IDH1 (0.31) IDH1
SCHEMBL6293531 0.85
SCHEMBL2822020 0.85 IDH1 (0.31) IDH1PTGDR2
SCHEMBL2822017 0.85 IDH1 (0.31) IDH1PTGDR2
SCHEMBL2818413 0.85 IDH1 (0.31) IDH1PTGDR2
SCHEMBL2818416 0.85 IDH1 (0.31) IDH1PTGDR2
SCHEMBL5672726 0.84 HDAC1 (0.34) IDH1PTGDR2
SCHEMBL5229789 0.83 IDH1 (0.34) IDH1PTGDR2
SCHEMBL5229785 0.83 IDH1 (0.34) IDH1PTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150980-B1 16-HALOGEN-EPOTHILONE DERIVATIVES, METHOD FOR PRODUCING THEM AND THEIR PHARMACEUTICAL USE BAYER SCHERING PHARMA AG (DE) 2007-08-22 EP disclosed
US-20050187270-A1 16-Halogen-epothilone derivatives, method for producing them and their pharmaceutical use BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2005-08-25 US disclosed
US-6610736-B1 Antitumor SCHERING AG (DE) 2003-08-26 US disclosed
EP-1150980-A2 16-HALOGEN-EPOTHILONE DERIVATIVES, METHOD FOR PRODUCING THEM AND THEIR PHARMACEUTICAL USE SCHERING AKTIENGESELLSCHAFT (DE) 2001-11-07 EP disclosed
WO-2000049021-A2 16-HALOGEN-EPOTHILONE DERIVATIVES, METHOD FOR PRODUCING THEM AND THEIR PHARMACEUTICAL USE SCHERING AKTIENGESELLSCHAFT (DE) 2000-08-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050187270-A1 16-Halogen-epothilone derivatives, method for producing them and their pharmaceutical use ABCB1, UGT2B17, CYP7B1 IDH1 2355/4885PTGDR2 539/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.