SCHEMBL5229724

SCHEMBL5229724

CCCn1c(=O)nc(SC)c2[nH]c(-c3cccnc3)nc21

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
TSHR P16473 1/20 0.52
ADORA2B P29275 9/20 0.50
ADORA2A P29274 6/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
KMT2A Q03164 1/20 0.50
HSD17B10 Q99714 1/20 0.50
ADORA1 P30542 4/20 0.48
ADORA3 P0DMS8 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230505 0.81 ADORA2B (0.66) ALDH1A1ADORA2BADORA2AKDM4EMEN1
SCHEMBL30682457 0.75 ADORA2B (0.70) ALDH1A1TSHRADORA2BADORA2AKDM4E
SCHEMBL30682506 0.75 ADORA2B (0.70) ALDH1A1TSHRADORA2BADORA2AKDM4E
SCHEMBL14345858 0.74 ADORA2B (0.58) ALDH1A1TSHRADORA2BADORA2AKDM4E
SCHEMBL30682533 0.73 ADORA2A (0.80) ALDH1A1TSHRADORA2BADORA2AKDM4E
SCHEMBL30682536 0.73 ADORA2A (0.80) ALDH1A1TSHRADORA2BADORA2AKDM4E
SCHEMBL30682607 0.72 ADORA2B (0.61) ALDH1A1TSHRADORA2BADORA2AKDM4E
SCHEMBL6092448 0.72 POLB (0.48) ADORA2BADORA2AADORA1
SCHEMBL6093879 0.71 ADORA1 (0.39) ADORA2BADORA2AADORA1ADORA3
SCHEMBL6093117 0.71 PDE2A (0.44) ADORA2BADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1092435-B1 REMEDIES FOR DIABETES KYOWA HAKKO KOGYO KK (JP) 2007-04-04 EP disclosed
US-6489331-B1 A CONDENSED PURINE DERIVATIVE AS AN ACTIVE INGREDIENT AS AN ENHANCER OF INSULIN SECRETION AND A MEDICAMENT FOR THE TREATMENT OF DIABETES KYOWA HAKKO KOGYO CO., LTD. (JP) 2002-12-03 US disclosed
EP-1092435-A1 REMEDIES FOR DIABETES KYOWA HAKKO KOGYO CO., LTD. (JP) 2001-04-18 EP disclosed