SCHEMBL5235220

SCHEMBL5235220

O=C1CCCN1N=C(Cc1ccnc2ccccc12)c1cccc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.44
CNR2 P34972 1/20 0.39
FLT1 P17948 2/20 0.39
MGLL Q99685 1/20 0.39
TACR1 P25103 1/20 0.38
CRHR1 P34998 1/20 0.38
DGAT2 Q96PD7 1/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
DRD2 P14416 1/20 0.36
DRD5 P21918 1/20 0.36
DRD3 P35462 1/20 0.36
PDGFRB P09619 1/20 0.36
CTSD P07339 1/20 0.36
BACE1 P56817 1/20 0.36
BACE2 Q9Y5Z0 1/20 0.36
CYP1A2 P05177 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5235216 1.00 KDR (0.44) KDRCNR2FLT1MGLLTACR1
SCHEMBL5233927 0.90 KDR (0.38) KDRCNR2FLT1TACR1DGAT2
SCHEMBL5233924 0.90 KDR (0.38) KDRCNR2FLT1TACR1DGAT2
SCHEMBL5239591 0.88 AR (0.39) KDRGAARAB9ALMNADRD2
SCHEMBL5239587 0.88 AR (0.39) KDRGAARAB9ALMNADRD2
SCHEMBL5238033 0.86 MGLL (0.41) KDRMGLLPOLBCYP1A2BRAF
SCHEMBL5238037 0.86 MGLL (0.41) KDRMGLLPOLBCYP1A2BRAF
SCHEMBL5240230 0.86 CYP1A2 (0.45) TACR1GAARAB9ALMNAPOLB
SCHEMBL5240236 0.86 CYP1A2 (0.45) TACR1GAARAB9ALMNAPOLB
SCHEMBL5238619 0.85 KDR (0.35) KDRMGLLTACR1HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed