SCHEMBL5235960

SCHEMBL5235960

COc1ccc(-c2ccc(S(C)(=O)=O)cc2)c(CC(=O)O)c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.54
PTGS2 P35354 6/20 0.53
MMP2 P08253 3/20 0.52
MMP8 P22894 3/20 0.52
MMP12 P39900 3/20 0.52
MMP13 P45452 3/20 0.52
MMP14 P50281 3/20 0.52
MMP16 P51512 3/20 0.52
MMP9 P14780 2/20 0.52
MMP1 P03956 1/20 0.52
MMP3 P08254 1/20 0.52
PTGS1 P23219 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.47
KDM4E B2RXH2 1/20 0.45
LCK P06239 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3738351 0.87 HSD17B10 (0.64) HSD17B10MMP2MMP8MMP12MMP13
SCHEMBL3735319 0.83 HSD17B10 (0.59) HSD17B10MMP2MMP8MMP12MMP13
SCHEMBL9890648 0.83 HSD17B10 (0.62) HSD17B10MMP2MMP8MMP12MMP13
SCHEMBL3736235 0.82 HSD17B10 (0.57) HSD17B10PTGS1SMN1; SMN2KDM4ELCK
SCHEMBL3738751 0.80 HSD17B10 (0.57) HSD17B10MMP2MMP12MMP9PTGS1
SCHEMBL8603589 0.79 PTGDR2 (0.57) PTGS2MMP2MMP8MMP12MMP13
SCHEMBL3740107 0.78 CYP1A2 (0.51) HSD17B10MMP2MMP8MMP12MMP13
SCHEMBL11889771 0.77 HSD17B10 (0.55) HSD17B10MMP2MMP8MMP12MMP13
SCHEMBL3749551 0.77 HSD17B10 (0.54) HSD17B10PTGS2MMP2MMP8MMP12
SCHEMBL15703754 0.77 MEN1 (0.55) HSD17B10MMP2MMP8MMP12MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1817031-A1 NOVEL SPECIFIC CASPASE-10 INHIBITORS Merck Patent GmbH (DE) 2007-08-15 EP claimed
WO-2006058592-A1 NOVEL SPECIFIC CASPASE-10 INHIBITORS MERCK PATENT GMBH (DE) 2006-06-08 WO claimed