SCHEMBL5236531

SCHEMBL5236531

O=C1CCCC(=O)N1/N=C(\Cc1ccnc2ccccc12)c1ccccn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.36
ALDH1A1 P00352 3/20 0.34
HTT P42858 1/20 0.34
BCHE P06276 1/20 0.34
LMNA P02545 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
KDM4E B2RXH2 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
FAAH O00519 1/20 0.34
MAPK9 P45984 1/20 0.33
RAB9A P51151 2/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
NAPRT Q6XQN6 1/20 0.33
P4HTM Q9NXG6 1/20 0.33
GAA P10253 2/20 0.32
MAPT P10636 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5236537 1.00 CYP1A2 (0.42) CYP1A2LOXL2ALDH1A1HTTBCHE
SCHEMBL5239257 0.88 CYP1A2 (0.41) CYP1A2LOXL2ALDH1A1HTTBCHE
SCHEMBL5239266 0.88 CYP1A2 (0.41) CYP1A2LOXL2ALDH1A1HTTBCHE
SCHEMBL5235695 0.79 CYP1A2 (0.38) CYP1A2LOXL2ALDH1A1HTTLMNA
SCHEMBL5235700 0.79 CYP1A2 (0.38) CYP1A2LOXL2ALDH1A1HTTLMNA
SCHEMBL5238516 0.78 CYP1A2 (0.41) CYP1A2LOXL2ALDH1A1HTTBCHE
SCHEMBL5238518 0.78 CYP1A2 (0.41) CYP1A2LOXL2ALDH1A1HTTBCHE
SCHEMBL5238497 0.78 GRM5 (0.34) CYP1A2ALDH1A1LMNASMN1; SMN2NPSR1
SCHEMBL5238502 0.78 GRM5 (0.34) CYP1A2ALDH1A1LMNASMN1; SMN2NPSR1
SCHEMBL5234873 0.77 CYP1A2 (0.39) CYP1A2LOXL2ALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed