SCHEMBL5238518

SCHEMBL5238518

CC1CC(=O)N(N=C(Cc2ccnc3ccccc23)c2ccccn2)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.41
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
FAAH O00519 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
HSD11B1 P28845 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
XIAP P98170 1/20 0.32
PDE4A P27815 1/20 0.32
BCHE P06276 1/20 0.32
GAA P10253 2/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
P2RX7 Q99572 1/20 0.31
IGF1R P08069 1/20 0.31
TACR1 P25103 1/20 0.31
PDK1 Q15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5238516 1.00 CYP1A2 (0.41) CYP1A2ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL5317558 0.86 CYP1A2 (0.39) CYP1A2ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL5276644 0.85 CYP1A2 (0.38) CYP1A2KDM4ESMN1; SMN2BCHEMAPT
SCHEMBL5276651 0.85 CYP1A2 (0.38) CYP1A2KDM4ESMN1; SMN2BCHEMAPT
SCHEMBL5235444 0.83 CYP1A2 (0.35) CYP1A2ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL5235435 0.83 CYP1A2 (0.35) CYP1A2ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL5239266 0.81 CYP1A2 (0.41) CYP1A2ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL5239257 0.81 CYP1A2 (0.41) CYP1A2ALDH1A1KDM4ELMNASMN1; SMN2
SCHEMBL6102141 0.81 ADRA1A (0.39) ALDH1A1SMN1; SMN2NPSR1MAPTHTT
SCHEMBL6102131 0.81 ADRA1A (0.39) ALDH1A1SMN1; SMN2NPSR1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397364-B1 NOVEL PYRROLE DERIVATIVES AS PHARMACEUTICAL AGENTS LILLY CO ELI (US) 2007-07-25 EP disclosed