SCHEMBL5239085

SCHEMBL5239085

O=C(O)c1ccc2c(c1)C=CNC2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.50
ALDH1A1 P00352 4/20 0.44
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA4 P22748 2/20 0.41
CA9 Q16790 2/20 0.41
TDP2 O95551 2/20 0.41
SRD5A2 P31213 4/20 0.40
MAPK1 P28482 2/20 0.40
KDM4E B2RXH2 5/20 0.39
HPGD P15428 1/20 0.39
ENPP2 Q13822 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 4/20 0.38
POLB P06746 2/20 0.37
GAA P10253 1/20 0.37
CA6 P23280 1/20 0.37
PTGS2 P35354 1/20 0.37
CA7 P43166 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23304599 0.85 PARP1 (0.44) PARP1ALDH1A1TDP2KDM4EHSD17B10
Hydrochloric Acid SCHEMBL7007714 0.83 PARP1 (0.47) PARP1ALDH1A1TDP2KDM4EHSD17B10
SCHEMBL30924717 0.82 HDAC6 (0.42) PARP1KDM4E
Hydrochloric Acid SCHEMBL7003754 0.80 PARP1 (0.44) PARP1ALDH1A1CA1CA2CA9
SCHEMBL7009677 0.79 NPC1 (0.50) PARP1ALDH1A1HPGDMAPTPOLB
SCHEMBL7004442 0.76 PARP1 (0.42) PARP1ALDH1A1CA12CA1CA2
Oxalic Acid SCHEMBL21489558 0.75 PARP1 (0.75) PARP1ALDH1A1SRD5A2KDM4EMAPT
Oxalic Acid SCHEMBL29882919 0.75 PARP1 (0.75) PARP1ALDH1A1SRD5A2KDM4EMAPT
SCHEMBL2115451 0.75 PARP1 (0.44) PARP1ALDH1A1KDM4EHSD17B10TSHR
Hydrochloric Acid SCHEMBL7001774 0.74 PARP1 (0.45) PARP1ALDH1A1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106831576-A Preparation method of 2-methyl-1-oxo-1, 2-dihydroisoquinoline-6-formic acid 北京六合宁远科技有限公司 2017-06-13 CN claimed
CN-106831576-A Preparation method of 2-methyl-1-oxo-1, 2-dihydroisoquinoline-6-formic acid 北京六合宁远科技有限公司 2017-06-13 CN disclosed
CN-102695708-B N1-pyrazolospiroketone acetyl-coA carboxylase inhibitors PFIZER INC. (US) 2014-10-15 CN disclosed
CN-102695708-A N1-pyrazolospiroketone acetyl-coA carboxylase inhibitors PFIZER 2012-09-26 CN disclosed
EP-1355886-B1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA PHARMACEUTICAL (JP) 2007-07-11 EP disclosed
EP-1399444-A2 NOVEL HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS Aventis Pharma S.A. (FR) 2004-03-24 EP disclosed
EP-1355886-A1 FUSED HETEROCYCLIC COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2003-10-29 EP disclosed
WO-2002100860-A2 HETEROCYCLIC COMPOUNDS, METHOD FOR PREPARING SAME AND USE THEREOF AS MEDICINES, IN PARTICULAR AS ANTI-BACTERIAL AGENTS AVENTIS PHARMA S.A. (FR) 2002-12-19 WO disclosed
WO-2002062764-A1 FUSED HETEROCYCLIC COMPOUNDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-08-15 WO disclosed