SCHEMBL23304599

SCHEMBL23304599

NC(=O)c1ccc2c(c1)C=CNC2

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 6/20 0.44
TSHR P16473 1/20 0.41
KDM1A O60341 2/20 0.38
LCK P06239 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HSD17B10 Q99714 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
MAPKAPK2 P49137 1/20 0.35
HSD17B3 P37058 1/20 0.34
TDP2 O95551 1/20 0.33
PRF1 P14222 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7007714 0.98 PARP1 (0.47) PARP1TSHRKDM1ALCKKDM4E
SCHEMBL2115451 0.87 PARP1 (0.44) PARP1TSHRKDM1ALCKKDM4E
SCHEMBL5239085 0.85 PARP1 (0.50) PARP1TSHRKDM1AKDM4EALDH1A1
Hydrochloric Acid SCHEMBL7003754 0.81 PARP1 (0.44) PARP1KDM4EALDH1A1
SCHEMBL30924717 0.81 HDAC6 (0.42) PARP1KDM4E
SCHEMBL7009677 0.75 NPC1 (0.50) PARP1ALDH1A1
SCHEMBL7094259 0.74 PARP1 (0.39) PARP1
SCHEMBL784887 0.74 KDM1A (0.41) PARP1TSHRKDM1ALCKKDM4E
SCHEMBL16229535 0.73 PARP1 (0.52) PARP1KDM4EALDH1A1TDP2
SCHEMBL23387607 0.73 PARP1 (0.52) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021086879-A1 COMPOUNDS AND METHODS OF USE TANGO THERAPEUTICS, INC. (US) 2021-05-06 WO disclosed