SCHEMBL5240243

SCHEMBL5240243

O=C(CC1CCCC1)C(O)(c1ccccc1)N1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.45
EPHX2 P34913 2/20 0.44
CHRM2 P08172 9/20 0.43
CHRM1 P11229 9/20 0.43
CHRM3 P20309 9/20 0.43
CYP2D6 P10635 3/20 0.43
KCNH2 Q12809 2/20 0.43
CHRM4 P08173 2/20 0.43
CHRM5 P08912 2/20 0.43
GRIN2D O15399 1/20 0.43
GRIN3B O60391 1/20 0.43
HRH1 P35367 1/20 0.43
GRIN1 Q05586 1/20 0.43
GRIN2A Q12879 1/20 0.43
GRIN2B Q13224 1/20 0.43
GRIN2C Q14957 1/20 0.43
GRIN3A Q8TCU5 1/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5240516 0.99 CCR1 (0.43) CCR1EPHX2CHRM2CHRM1CHRM3
SCHEMBL3981459 0.82 CHRM3 (0.49) CHRM2CHRM1CHRM3TSHR
SCHEMBL2763733 0.73 CHRM3 (0.41) CCR1CHRM2CHRM1CHRM3CYP2D6
SCHEMBL5999930 0.71 EPHX2 (0.45) CCR1EPHX2CHRM2CHRM1CHRM3
SCHEMBL2796932 0.69 CHRM3 (0.40) CCR1CHRM2CHRM1CHRM3CYP2D6
SCHEMBL4618235 0.68 KEAP1 (0.53) CCR1EPHX2CHRM2CHRM1CHRM3
SCHEMBL13116345 0.68 KEAP1 (0.53) CCR1EPHX2CHRM2CHRM1CHRM3
SCHEMBL7569557 0.68 KEAP1 (0.53) CHRM2CHRM1CHRM3CYP2D6KCNH2
Hydrochloric Acid SCHEMBL7433430 0.68 CHRM2 (0.43) CHRM2CHRM1CHRM3CYP2D6KCNH2
SCHEMBL4887507 0.67 HTT (0.60) CHRM2CHRM1CHRM3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794161-A2 MUSCARINIC RECEPTOR ANTAGONISTS Ranbaxy Laboratories Limited (IN) 2007-06-13 EP disclosed
WO-2006032994-A2 MUSCARINIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2006-03-30 WO disclosed