SCHEMBL5243233

SCHEMBL5243233

COC(CC(N)c1cccs1)OC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.36
GNRHR P30968 1/20 0.34
SLC6A2 P23975 4/20 0.33
SLC6A4 P31645 4/20 0.33
SLC6A3 Q01959 3/20 0.33
HSD17B2 P37059 1/20 0.32
CNR2 P34972 1/20 0.32
CES2 O00748 1/20 0.32
CES1 P23141 1/20 0.32
KEAP1 Q14145 1/20 0.32
SLC7A5 Q01650 1/20 0.31
HTR1A P08908 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MLNR O43193 1/20 0.31
CACNA1F O60840 1/20 0.31
CYP1A2 P05177 1/20 0.31
ADRB1 P08588 1/20 0.31
CYP3A4 P08684 1/20 0.31
GAA P10253 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15765746 0.79 ALOX5 (0.42) ALOX5SLC6A2SLC6A4SLC6A3CES2
SCHEMBL12262736 0.78 ALOX5 (0.38) ALOX5GNRHRSLC6A2SLC6A4SLC6A3
SCHEMBL1888261 0.75
SCHEMBL12261602 0.75
SCHEMBL3465862 0.75
SCHEMBL14511482 0.75
SCHEMBL5168943 0.74 ALOX5 (0.41) ALOX5SLC6A2SLC6A4SLC6A3CES2
SCHEMBL14445287 0.73 CYP2C19 (0.40) ALOX5HSD17B2CES2CES1KEAP1
Hydrochloric Acid SCHEMBL15476689 0.73 ALOX5 (0.40) ALOX5SLC6A2SLC6A4SLC6A3CES2
Hydrochloric Acid SCHEMBL4472643 0.73 ALOX5 (0.40) ALOX5SLC6A2SLC6A4SLC6A3CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833797-A1 AZACYCLIC COMPOUNDS AS INHBITORS OF SENSORY NEURONE SPECIFIC CHANNELS (SNS) VERNALIS (R&D) LTD (GB) 2007-09-19 EP disclosed
WO-2006082354-A1 AZACYCLIC COMPOUNDS AS INHIBITORS OF SENSORY NEURONE SPECIFIC CHANNELS ( SNS ) VERNALIS (R & D) LIMITED (GB) 2006-08-10 WO disclosed