SCHEMBL5246381

SCHEMBL5246381

CC(C1CCNC1)N(C)c1nc2c(C(N)=O)c[c]cc2s1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 10/20 0.34
IRAK4 Q9NWZ3 7/20 0.32
PARP2 Q9UGN5 1/20 0.31
PIM1 P11309 3/20 0.30
KCNH2 Q12809 3/20 0.30
PIM2 Q9P1W9 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5244562 0.91 PARP1 (0.33) PARP1IRAK4PARP2PIM1KCNH2
SCHEMBL5248275 0.90 PARP1 (0.33) PARP1PARP2
SCHEMBL5245345 0.89 PARP1 (0.32) PARP1IRAK4
SCHEMBL3750058 0.80 PARP14 (0.34) PARP1
SCHEMBL3749075 0.80 PARP1 (0.34) PARP1IRAK4PARP2
SCHEMBL3749097 0.71 PARP1 (0.38) PARP1PARP2
SCHEMBL3750053 0.69 PARP1 (0.35) PARP1PARP2
SCHEMBL3751235 0.69 PARP1 (0.39) PARP1PARP2
SCHEMBL3756206 0.68 PARP1 (0.36) PARP1IRAK4PARP2
SCHEMBL3746699 0.68 PARP1 (0.40) PARP1IRAK4PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1828177-A2 NOVEL MCH RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2007-09-05 EP disclosed
WO-2006066173-A2 NOVEL MCH RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 2006-06-22 WO disclosed