SCHEMBL5247140

SCHEMBL5247140

O=C(O)[C@H]1CCCN(c2nc(Nc3ccccn3)c3c(cnn3CCOCC(F)(F)F)n2)C1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 19/20 0.49
KCNH2 Q12809 5/20 0.42
IDH2 P48735 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5245602 1.00 PDE5A (0.49) PDE5AKCNH2IDH2
SCHEMBL5247942 0.96 PDE5A (0.51) PDE5AKCNH2
SCHEMBL5245416 0.91 PDE5A (0.53) PDE5AKCNH2IDH2
SCHEMBL5246388 0.91 PDE5A (0.53) PDE5AKCNH2
SCHEMBL5247705 0.89 PDE5A (0.44) PDE5AKCNH2IDH2
SCHEMBL5284677 0.87 PDE5A (0.59) PDE5AKCNH2
SCHEMBL5244271 0.87 PDE5A (0.55) PDE5AKCNH2
SCHEMBL5247381 0.87 PDE5A (0.55) PDE5AKCNH2
SCHEMBL5247815 0.86 PDE5A (0.59) PDE5AKCNH2
SCHEMBL5325370 0.86 PDE5A (0.59) PDE5AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809632-A2 PYRAZOLO[4,3-D]PYRIMIDINE DERIVATIVES USEFUL AS PDE-5 INHIBITORS Pharmacia & Upjohn Company LLC (US) 2007-07-25 EP disclosed
WO-2006046135-A2 PYRAZOLO[4,3-D] PYRIMIDINE DERIVATIVES USEFUL AS PDE-5 INHIBITORS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-05-04 WO disclosed