SCHEMBL5248396

SCHEMBL5248396

BrCCc1ccc2nccnc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ECE2 P0DPD6 1/20 0.42
SHMT2 P34897 1/20 0.41
TDP1 Q9NUW8 2/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
L3MBTL1 Q9Y468 1/20 0.35
MET P08581 1/20 0.35
MAPT P10636 1/20 0.34
HDAC3 O15379 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34
HDAC4 P56524 1/20 0.34
TUBA1B P68363 1/20 0.34
TUBA4A P68366 1/20 0.34
TUBB4B P68371 1/20 0.34
TUBB3 Q13509 1/20 0.34
HDAC1 Q13547 1/20 0.34
TUBB2A Q13885 1/20 0.34
TUBB8 Q3ZCM7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31287240 1.00 ECE2 (0.42) ECE2SHMT2TDP1NPC1RAB9A
SCHEMBL4280865 0.88 ECE2 (0.41) ECE2SHMT2TDP1NPC1RAB9A
Bromide SCHEMBL4280985 0.86 ECE2 (0.40) ECE2SHMT2TDP1NPC1RAB9A
SCHEMBL843959 0.83 ECE2 (0.45) ECE2SHMT2TDP1NPC1RAB9A
SCHEMBL6851853 0.79 ECE2 (0.42) ECE2SHMT2TDP1NPC1RAB9A
SCHEMBL9971308 0.79 CNR1 (0.44) ECE2SHMT2NPC1RAB9AMAPT
SCHEMBL5155836 0.79 KDM4E (0.47) ECE2SHMT2TDP1NPC1RAB9A
SCHEMBL2859216 0.79 TAAR1 (0.45) ECE2SHMT2TDP1L3MBTL1MAPT
SCHEMBL5151371 0.79 ECE2 (0.42) ECE2SHMT2TDP1NPC1RAB9A
SCHEMBL31287242 0.79 KDM4E (0.47) ECE2SHMT2TDP1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1968948-A Process for preparing gonadotropin releasing hormone receptor antagonists WYETH CORP (US) 2007-05-23 CN claimed
CN-102775396-B Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-08 CN disclosed
CN-102775396-A Modulators of ATP-binding cassette transporters VERTEX PHARMA 2012-11-14 CN disclosed
CN-101356170-B Heterocyclic modulators of ATP-binding cassette transporters VERTEX PHARMA 2012-09-26 CN disclosed
CN-101356170-A Heterocyclic modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2009-01-28 CN disclosed
CN-101006078-A Gonadotropin releasing hormone receptor antagonists WYETH CORP (US) 2007-07-25 CN disclosed
CN-1968948-A Process for preparing gonadotropin releasing hormone receptor antagonists WYETH CORP (US) 2007-05-23 CN disclosed
EP-1758895-A1 GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONISTS Wyeth a Corporation of the State of Delaware (US) 2007-03-07 EP disclosed
CN-1256326-C Novel 4- (oxoxyphenyl) -3-oxopiperidines for the treatment of cardiac and renal insufficiency HOFFMANN LA ROCHE (CH) 2006-05-17 CN disclosed
WO-2006009734-A1 GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONISTS WYETH (US) 2006-01-26 WO disclosed
CN-1202152-A Novel 4- (oxoxyphenyl) -3-oxopiperidines for the treatment of cardiac and renal insufficiency HOFFMANN LA ROCHE (CH) 1998-12-16 CN disclosed
CN-1031266-C Process for preparation of heterocycle ether derivatives ZENECA LTD (GB) 1996-03-13 CN disclosed
CN-1046903-A Process for preparing heterocyclic ether derivatives ICI PLC (GB) 1990-11-14 CN disclosed