SCHEMBL2859216

SCHEMBL2859216

NCCc1ccc2nccnc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 10/20 0.45
KDM4E B2RXH2 4/20 0.45
ADRA2A P08913 3/20 0.45
SLC6A2 P23975 3/20 0.45
MAPT P10636 2/20 0.45
DRD2 P14416 2/20 0.45
DRD1 P21728 2/20 0.45
DRD4 P21917 2/20 0.45
DRD5 P21918 2/20 0.45
MAPK1 P28482 2/20 0.45
DRD3 P35462 2/20 0.45
RECQL P46063 2/20 0.45
SLC6A3 Q01959 2/20 0.45
TDP1 Q9NUW8 2/20 0.45
ALDH1A1 P00352 2/20 0.45
HTR1A P08908 2/20 0.45
PNMT P11086 1/20 0.45
TP53 P04637 1/20 0.45
ADRB2 P07550 1/20 0.45
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2860410 0.83 LOXL2 (0.47) ADRB2SHMT2LOXL2ECE2
SCHEMBL31367022 0.83 LOXL2 (0.47) ADRB2SHMT2LOXL2ECE2
Hydrochloric Acid SCHEMBL28952754 0.81 LOXL2 (0.45) ADRB2SHMT2LOXL2GAAECE2
SCHEMBL5155836 0.79 KDM4E (0.47) KDM4EMAPTTDP1ALDH1A1CYP2D6
SCHEMBL31287240 0.79 ECE2 (0.42) KDM4EADRA2AMAPTTDP1CYP2D6
SCHEMBL31287242 0.79 KDM4E (0.47) KDM4EMAPTTDP1ALDH1A1CYP2D6
SCHEMBL5248396 0.79 ECE2 (0.42) KDM4EADRA2AMAPTTDP1CYP2D6
SCHEMBL6851853 0.79 ECE2 (0.42) KDM4EADRA2AMAPTTDP1ALDH1A1
SCHEMBL9971308 0.79 CNR1 (0.44) MAPTCYP2D6SHMT2GAAECE2
SCHEMBL5151371 0.79 ECE2 (0.42) ADRA2AMAPTTDP1CYP2D6SHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139334-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF Renovis, Inc. (US) 2010-01-06 EP disclosed
WO-2008130481-A1 2-CYANOPHENYL FUSED HETEROCYCLIC COMPOUNDS, AND COMPOSITIONS AND USES THEREOF RENOVIS, INC. (US) 2008-10-30 WO disclosed