SCHEMBL5249146

SCHEMBL5249146

O=C(NCC(F)(F)F)c1ccc(-n2nnc(C(=O)NCc3cccc(Cl)c3)c2COCc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.51
ABCB1 P08183 1/20 0.43
PTGER1 P34995 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C19 P33261 2/20 0.41
NPC1 O15118 1/20 0.41
CYP2C9 P11712 1/20 0.41
RAB9A P51151 1/20 0.41
POLB P06746 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
PTGER4 P35408 1/20 0.41
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MMP13 P45452 1/20 0.40
CXCR3 P49682 1/20 0.40
PLA2G1B P04054 1/20 0.39
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5250048 0.92 EPHX2 (0.46) CCR1RAB9AMEN1KMT2A
SCHEMBL5246087 0.91 CCR1 (0.47) CCR1ABCB1PTGER1MEN1KMT2A
SCHEMBL5248465 0.91 CCR1 (0.46) CCR1ABCB1MEN1KMT2AHTT
SCHEMBL5245586 0.91 CCR1 (0.46) CCR1MEN1KMT2APTGER4MAPT
SCHEMBL5247796 0.90 CCR1 (0.45) CCR1ABCB1CYP1A2CYP2D6CYP2C19
SCHEMBL5249014 0.90 CCR1 (0.45) CCR1ABCB1MEN1KMT2APTGER4
SCHEMBL5244716 0.90 CCR1 (0.57) CCR1CYP1A2CYP2D6CYP2C19RAB9A
SCHEMBL5244866 0.89 CCR1 (0.44) CCR1ABCB1POLBMEN1KMT2A
SCHEMBL5247606 0.89 MAPK14 (0.54) CCR1ABCB1
SCHEMBL5246577 0.89 SMN1; SMN2 (0.47) CCR1CYP2D6CYP2C9POLBPTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1867331-A1 TRIAZOLE DERIVATIVE AND THE USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2007-12-19 EP disclosed