SCHEMBL5250675

SCHEMBL5250675

CC1CCCC(C)N1S(=O)(=O)c1ccc(Cl)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACHE P22303 7/20 1.00
PSEN1 P49768 7/20 1.00
PSEN2 P49810 7/20 1.00
APH1B Q8WW43 7/20 1.00
NCSTN Q92542 7/20 1.00
APH1A Q96BI3 7/20 1.00
PSENEN Q9NZ42 7/20 1.00
POLB P06746 2/20 0.60
AKR1C3 P42330 1/20 0.57
LMNA P02545 1/20 0.57
KMT2A Q03164 3/20 0.53
MEN1 O00255 2/20 0.53
ALDH1A1 P00352 1/20 0.50
TP53 P04637 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5915359 1.00 ACHE (1.00) ACHEPSEN1PSEN2APH1BNCSTN
SCHEMBL5915351 0.93 ACHE (0.87) ACHEPSEN1PSEN2APH1BNCSTN
SCHEMBL5915290 0.93 ACHE (0.87) ACHEPSEN1PSEN2APH1BNCSTN
SCHEMBL13248930 0.84 ACHE (1.00) ACHEPSEN1PSEN2APH1BNCSTN
SCHEMBL13069242 0.84 ACHE (1.00) ACHEPSEN1PSEN2APH1BNCSTN
SCHEMBL19392468 0.84 ACHE (1.00) ACHEPSEN1PSEN2APH1BNCSTN
SCHEMBL9144277 0.84 PSEN1 (0.72) ACHEPSEN1PSEN2APH1BNCSTN
SCHEMBL2221432 0.84 PSEN1 (0.72) ACHEPSEN1PSEN2APH1BNCSTN
SCHEMBL12793076 0.83 ACHE (0.73) ACHEPSEN1PSEN2APH1BNCSTN
SCHEMBL2220964 0.82 PSEN1 (0.70) ACHEPSEN1PSEN2APH1BNCSTN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1758884-A2 N-CYCLIC SULFONAMIDO INHIBITORS OF GAMMA SECRETASE Elan Pharmaceuticals, Inc. (US) 2007-03-07 EP claimed
EP-1758895-A1 GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONISTS Wyeth a Corporation of the State of Delaware (US) 2007-03-07 EP claimed
US-20060035884-A1 N-cyclic sulfonamido inhibitors of gamma secretase ELAN PHARMACEUTICALS, INC. (US) 2006-02-16 US claimed
WO-2006009734-A1 GONADOTROPIN RELEASING HORMONE RECEPTOR ANTAGONISTS WYETH (US) 2006-01-26 WO claimed
WO-2005113542-A2 N-CYCLIC SULFONAMIDO INHIBITORS OF GAMMA SECRETASE ELAN PHARMACEUTICALS, INC. (US) 2005-12-01 WO claimed
US-20060035884-A1 N-cyclic sulfonamido inhibitors of gamma secretase ELAN PHARMACEUTICALS, INC. (US) 2006-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035884-A1 N-cyclic sulfonamido inhibitors of gamma secretase BACE1, BACE2, APH1B ACHE 13/4885PSEN1 4/4885PSEN2 8/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.