SCHEMBL5250810

SCHEMBL5250810

CN(C)C(c1ccccc1)c1ncc(C(=O)NCc2ccccc2Cl)c(O)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 5/20 0.45
L3MBTL1 Q9Y468 3/20 0.45
HPGD P15428 3/20 0.45
HSD17B10 Q99714 3/20 0.45
MAPT P10636 2/20 0.44
PLA2G1B P04054 1/20 0.44
POLB P06746 1/20 0.44
ATG4B Q9Y4P1 1/20 0.44
MAPK8 P45983 2/20 0.44
LMNA P02545 4/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
THRB P10828 1/20 0.43
PKM P14618 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5123530 0.83 ALDH1A1 (0.46) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL3410324 0.69 MEN1 (0.49) ALDH1A1MEN1KMT2AKDM4EL3MBTL1
SCHEMBL5119574 0.68 TACR1 (0.46) ALDH1A1MEN1KMT2AMAPTCYP1A2
SCHEMBL11000305 0.68 KDM4E (0.33) ALDH1A1MEN1KMT2AKDM4EMAPT
SCHEMBL6643772 0.67 ALDH1A1 (0.46) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL5123821 0.67 MAOB (0.45) ALDH1A1MEN1KMT2AKDM4EHPGD
SCHEMBL15358460 0.67 HDAC3 (0.55) ALDH1A1MEN1KMT2AMAPTPLA2G1B
SCHEMBL5122580 0.66 MAOB (0.41) MEN1KMT2A
SCHEMBL6645608 0.65 ALDH1A1 (0.46) ALDH1A1KMT2AKDM4EL3MBTL1HPGD
SCHEMBL5121257 0.65 SMN1; SMN2 (0.43) ALDH1A1KMT2AKDM4EL3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1441734-B1 DIHYDROXYPYRIMIDINE CARBOXAMIDE INHIBITORS OF HIV INTEGRASE ANGELETTI P IST RICHERCHE BIO (IT) 2007-02-28 EP disclosed