SCHEMBL5253301

SCHEMBL5253301

COc1ccc2nccc([C@@H](O)CN3CC[CH]CC3)c2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.61
SLC2A1 P11166 8/20 0.59
CYP2D6 P10635 5/20 0.49
ALDH1A1 P00352 5/20 0.49
HSD17B10 Q99714 5/20 0.49
KDM4E B2RXH2 4/20 0.49
HPGD P15428 3/20 0.49
CYP3A4 P08684 3/20 0.49
TSHR P16473 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ADRA2A P08913 2/20 0.49
SLC6A4 P31645 2/20 0.49
OPRM1 P35372 2/20 0.49
SLC6A3 Q01959 2/20 0.49
CHRM2 P08172 1/20 0.49
LMNA P02545 1/20 0.47
THRB P10828 1/20 0.47
SLC22A1 O15245 1/20 0.47
ABCC4 O15439 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5253304 1.00 KCNH2 (0.61) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10
SCHEMBL13356470 0.91 SLC2A1 (0.59) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10
SCHEMBL13356412 0.91 SLC2A1 (0.59) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10
SCHEMBL5757621 0.89 NCF1 (0.58) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10
SCHEMBL6484670 0.89 NCF1 (0.58) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10
SCHEMBL6484668 0.89 NCF1 (0.58) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10
SCHEMBL4273370 0.88 SLC2A1 (0.59) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10
SCHEMBL4273361 0.88 SLC2A1 (0.59) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10
SCHEMBL4273379 0.88 SLC2A1 (0.59) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10
SCHEMBL4269291 0.87 SLC2A1 (0.63) KCNH2SLC2A1CYP2D6ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1359908-B1 QUINOLINES AND NITROGENATED DERIVATIVES THEREOF SUBSTITUTED IN 4-POSITION BY A PIPERIDINE-CONTAINING MOIETY AND THEIR USE AS ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM PLC (GB) 2007-08-22 EP claimed
EP-1359908-A1 QUINOLINES AND NITROGENATED DERIVATIVES THEREOF SUBSTITUTED IN 4-POSITION BY A PIPERIDINE-CONTAINING MOIETY AND THEIR USE AS ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM PLC (GB) 2003-11-12 EP disclosed
WO-2002056882-A1 QUINOLINES AND NITROGENATED DERIVAIVE THEREOF SUBSTITUTED IN 4-POSITION BY A PIPERIDINE-CONTAINING MOIETY AND THEIR USE AS ANTIBACTERIAL AGENTS SMITHKLINE BEECHAM P.L.C. (GB) 2002-07-25 WO disclosed