SCHEMBL5255284

SCHEMBL5255284

COc1cc(C2=C(c3cn(CCBr)c4ccccc34)C(=O)NC2=O)c2occc2c1

nearest known ligand 0.77

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 12/20 0.77
KDR P35968 6/20 0.49
FLT3 P36888 3/20 0.49
QPCT Q16769 1/20 0.49
PRKCA P17252 3/20 0.48
PRKACA P17612 2/20 0.46
PRKACG P22612 2/20 0.46
PRKACB P22694 2/20 0.46
CAMK2D Q13557 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4991182 0.95 GSK3B (0.75) GSK3BKDRFLT3QPCTPRKACA
SCHEMBL5257432 0.91 GSK3B (0.77) GSK3BKDRFLT3QPCTPRKCA
SCHEMBL5257465 0.90 GSK3B (0.75) GSK3BKDRFLT3QPCTPRKCA
SCHEMBL5258462 0.89 GSK3B (0.75) GSK3BKDRFLT3QPCTPRKCA
SCHEMBL4992178 0.89 GSK3B (0.75) GSK3BKDRFLT3QPCTPRKCA
SCHEMBL4994614 0.88 GSK3B (0.72) GSK3BKDRFLT3QPCTPRKCA
SCHEMBL5260235 0.87 GSK3B (1.00) GSK3BKDRFLT3QPCTPRKCA
SCHEMBL4984745 0.87 GSK3B (0.70) GSK3BKDRPRKCA
SCHEMBL5256402 0.82 GSK3B (0.65) GSK3BKDRPRKCA
SCHEMBL4991290 0.78 GSK3B (0.62) GSK3BFLT3PRKCAPRKACAPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487822-B1 PYRROLE-2,5-DIONE DERIVATIVES AND THEIR USE AS GSK-3 INHIBITORS LILLY CO ELI (US) 2007-08-01 EP disclosed
CN-1639152-A Pyrrole-2, 5-dione derivatives and their use as GSK-3 inhibitors LILLY CO ELI (US) 2005-07-13 CN disclosed