SCHEMBL5256402

SCHEMBL5256402

COc1cc(C2=C(c3cn(C(C)C)c4ccccc34)C(=O)NC2=O)c2occc2c1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 7/20 0.65
PRKCA P17252 7/20 0.48
PRKCB P05771 2/20 0.46
PRKCH P24723 1/20 0.46
PRKCE Q02156 1/20 0.46
PRKCQ Q04759 1/20 0.46
PRKCD Q05655 1/20 0.46
CDK2 P24941 2/20 0.42
CCNE2 O96020 1/20 0.42
CDK4 P11802 1/20 0.42
CCND1 P24385 1/20 0.42
CCNE1 P24864 1/20 0.42
MKNK1 Q9BUB5 1/20 0.42
MKNK2 Q9HBH9 1/20 0.42
KDR P35968 1/20 0.42
PRKCG P05129 1/20 0.42
CCNT1 O60563 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK9 P50750 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4984745 0.87 GSK3B (0.70) GSK3BPRKCACDK2CCNE2CDK4
SCHEMBL5257465 0.85 GSK3B (0.75) GSK3BPRKCAKDR
SCHEMBL5255284 0.82 GSK3B (0.77) GSK3BPRKCAKDR
SCHEMBL5257432 0.82 GSK3B (0.77) GSK3BPRKCAKDR
SCHEMBL4991182 0.81 GSK3B (0.75) GSK3BKDR
SCHEMBL4992178 0.81 GSK3B (0.75) GSK3BPRKCAPRKCBPRKCECDK4
SCHEMBL5258462 0.81 GSK3B (0.75) GSK3BPRKCAPRKCBPRKCHPRKCE
SCHEMBL4991290 0.80 GSK3B (0.62) GSK3BPRKCAPRKCBPRKCHPRKCE
SCHEMBL4994614 0.79 GSK3B (0.72) GSK3BPRKCAPRKCBPRKCHPRKCE
SCHEMBL5260235 0.79 GSK3B (1.00) GSK3BPRKCAPRKCBPRKCHPRKCE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1487822-B1 PYRROLE-2,5-DIONE DERIVATIVES AND THEIR USE AS GSK-3 INHIBITORS LILLY CO ELI (US) 2007-08-01 EP disclosed