SCHEMBL5256293

SCHEMBL5256293

N#CC(NC[C@H]1CCCC[C@@H]1NC(=O)c1cc2c(F)cc(F)cc2[nH]1)C1CC1

nearest known ligand 0.37

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.37
MLLT1 Q03111 1/20 0.37
CNR1 P21554 1/20 0.36
SLC2A1 P11166 1/20 0.35
PYGL P06737 1/20 0.30
HCRTR1 O43613 1/20 0.30
TAS1R3 Q7RTX0 1/20 0.30
TAS1R1 Q7RTX1 1/20 0.30
TAS1R2 Q8TE23 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5254517 0.86 MLLT1 (0.55) GHSRMLLT1CNR1PYGL
SCHEMBL6840849 0.83 GHSR (0.38) GHSRMLLT1CNR1SLC2A1
SCHEMBL5256296 0.83 GHSR (0.38) GHSRMLLT1CNR1SLC2A1
SCHEMBL5260386 0.81 HDAC3 (0.41) HCRTR1
SCHEMBL5255164 0.81 KDM4E (0.44) PYGL
SCHEMBL5256290 0.80 GHSR (0.37) GHSRMLLT1CNR1SLC2A1PYGL
SCHEMBL5261818 0.79 KMT2A (0.47)
SCHEMBL5254550 0.79 MLLT1 (0.41) MLLT1PYGL
SCHEMBL5257320 0.79 F10 (0.48) PYGL
SCHEMBL5257173 0.79 MLLT1 (0.41) MLLT1PYGL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453801-B1 SUBSTITUTED 2-AMINO-CYCLOALKANECARBOXAMIDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed