SCHEMBL5257232

SCHEMBL5257232

N#CC(NC[C@H]1CCCC[C@@H]1NC(=O)c1ccc2cc[nH]c2c1)C1CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.47
F10 P00742 1/20 0.46
SMYD3 Q9H7B4 3/20 0.44
MAPK11 Q15759 1/20 0.41
MAPK14 Q16539 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
HTR3A P46098 1/20 0.41
ESR1 P03372 3/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 3/20 0.39
ENPP2 Q13822 1/20 0.39
MAPT P10636 2/20 0.38
ALOX12 P18054 1/20 0.38
CTSK P43235 1/20 0.37
HDAC1 Q13547 3/20 0.37
HDAC2 Q92769 3/20 0.37
HDAC3 O15379 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5256986 0.94 SMYD3 (0.45) CHRNA7F10SMYD3TAS1R3TAS1R1
SCHEMBL5258888 0.82 SSTR3 (0.38) F10TAS1R3TAS1R1KDM4EALDH1A1
SCHEMBL6834634 0.82 CHRNA7 (0.48) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL5257234 0.82 CHRNA7 (0.48) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL6834935 0.82 CHRNA7 (0.48) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL5257229 0.79 CHRNA7 (0.46) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL5255164 0.77 KDM4E (0.44) CHRNA7HTR3AKDM4EALDH1A1HPGD
SCHEMBL5257320 0.77 F10 (0.48) F10SMYD3
SCHEMBL5255593 0.77 DRD4 (0.36) F10KDM4EALDH1A1HPGDCTSK
SCHEMBL5254550 0.76 MLLT1 (0.41) F10SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453801-B1 SUBSTITUTED 2-AMINO-CYCLOALKANECARBOXAMIDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed