SCHEMBL6834634

SCHEMBL6834634

N#C[C@@H](NC(=O)[C@@H]1CCCCC1NC(=O)c1ccc2cc[nH]c2c1)C1CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.48
F10 P00742 2/20 0.46
SMYD3 Q9H7B4 2/20 0.42
MAPK11 Q15759 1/20 0.42
MAPK14 Q16539 1/20 0.42
TAS1R3 Q7RTX0 2/20 0.41
TAS1R1 Q7RTX1 2/20 0.41
HTR3A P46098 1/20 0.41
ESR1 P03372 3/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40
HSD17B10 Q99714 2/20 0.40
ENPP2 Q13822 1/20 0.40
CTSK P43235 1/20 0.38
KDM5A P29375 1/20 0.37
RXFP2 Q8WXD0 1/20 0.37
TACR1 P25103 1/20 0.36
MAPT P10636 1/20 0.36
ALOX12 P18054 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5257234 1.00 CHRNA7 (0.48) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL6834935 1.00 CHRNA7 (0.48) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL6838485 0.93 SMYD3 (0.43) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL5255323 0.93 SMYD3 (0.43) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL6840603 0.83 CTSK (0.47) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL6382169 0.82 TAS1R3 (0.54) TAS1R3TAS1R1CTSK
SCHEMBL6382172 0.82 TAS1R3 (0.54) TAS1R3TAS1R1CTSK
SCHEMBL5257232 0.82 CHRNA7 (0.47) CHRNA7F10SMYD3MAPK11MAPK14
SCHEMBL5345197 0.81 NPC1 (0.39) TAS1R3TAS1R1CTSK
SCHEMBL5260931 0.81 AKT1 (0.44) SMYD3MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6759428-B2 SUCH AS N-((1,2)-2-(((CYANO(CYCLOPROPYL)METHYL)AMINO)CARBONYL) CYCLOHEXYL)-1H-INDOLE-2-CARBOXAMIDE; CATHEPSIN K INHIBITORS ROCHE PALO ALTO LLC 2004-07-06 US disclosed