SCHEMBL5258357

SCHEMBL5258357

N#Cc1ccc(C(=O)NC2CN(C(c3ccc(Cl)cc3)c3ccc(Cl)cc3)CC2CO)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 2/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
SLC6A5 Q9Y345 1/20 0.43
EPHX2 P34913 2/20 0.42
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
CHRNA7 P36544 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CNR1 P21554 2/20 0.39
CNR2 P34972 1/20 0.39
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
NSD2 O96028 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2516280 1.00 SLC6A9 (0.43) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2
SCHEMBL15933111 0.89 SLC6A9 (0.41) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2
SCHEMBL2522593 0.88 CYP2C9 (0.40) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2
SCHEMBL15929802 0.85 SLC6A9 (0.38) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2
SCHEMBL2517127 0.83 EPHX2 (0.41) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2
SCHEMBL5255473 0.83 EPHX2 (0.41) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2
SCHEMBL5252394 0.82 TP53 (0.41) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2
SCHEMBL2516227 0.82 TP53 (0.41) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2
SCHEMBL2517186 0.82 TP53 (0.41) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2
SCHEMBL5250135 0.82 TP53 (0.41) SLC6A9CYP2D6CYP2C9SLC6A5EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1748980-A1 PYRROLIDINE DERIVATIVES AS CB1-RECEPTOR ANTAGONISTS TANABE SEIYAKU CO., LTD. (JP) 2007-02-07 EP disclosed
WO-2005115977-A1 PYRROLIDINE DERIVATIVES AS CB1-RECEPTOR ANTAGONISTS TANABE SEIYAKU CO., LTD. (JP) 2005-12-08 WO disclosed