SCHEMBL5258758

SCHEMBL5258758

Cc1nc(CC#CCc2ccccc2)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.36
KCNH2 Q12809 3/20 0.36
GRM5 P41594 2/20 0.36
RAB9A P51151 1/20 0.34
ADORA2A P29274 2/20 0.32
ADORA1 P30542 2/20 0.32
TAAR1 Q96RJ0 1/20 0.32
HAO1 Q9UJM8 1/20 0.31
FFAR1 O14842 1/20 0.30
FFAR4 Q5NUL3 1/20 0.30
ALDH1A1 P00352 2/20 0.30
HPGD P15428 1/20 0.30
GAA P10253 1/20 0.30
AKT1 P31749 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL82538 0.79 TAAR1 (0.43) RAB9AADORA2AADORA1TAAR1ALDH1A1
SCHEMBL11091944 0.77 KCNH2 (0.52) KCNH2RAB9ATAAR1ALDH1A1HPGD
Water SCHEMBL10981448 0.77 TAAR1 (0.42) RAB9AADORA2AADORA1TAAR1ALDH1A1
Methane SCHEMBL28186549 0.76 KCNH2 (0.50) KCNH2RAB9ATAAR1ALDH1A1HPGD
Fluoride SCHEMBL28059937 0.76 TAAR1 (0.41) RAB9AADORA2AADORA1TAAR1ALDH1A1
SCHEMBL5703443 0.72 GRM5 (0.51) DHFRKCNH2GRM5RAB9AALDH1A1
SCHEMBL3888886 0.71 CALM1 (0.50) KCNH2TAAR1FFAR1FFAR4ALDH1A1
SCHEMBL103845 0.70 GRM5 (0.60) KCNH2GRM5FFAR1FFAR4
SCHEMBL28094600 0.69 TAAR1 (0.53) ADORA2AADORA1TAAR1ALDH1A1HPGD
Trifluoroacetic Acid SCHEMBL28186507 0.68 KCNH2 (0.41) KCNH2GRM5FFAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765795-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS Addex Pharmaceuticals SA (CH) 2007-03-28 EP disclosed
WO-2005123703-A2 ALKYNYL DERIVATIVES AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS ADDEX PHARMACEUTICALS SA (CH) 2005-12-29 WO disclosed