SCHEMBL5261807

SCHEMBL5261807

CC(C)(C)OC(=O)Nc1ccc2[nH]c(C(=O)N[C@H]3CCCC[C@H]3C(=O)NC(C#N)C3CC3)cc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LEF1 Q9UJU2 1/20 0.46
MLLT1 Q03111 1/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
PYGL P06737 3/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
KDM4E B2RXH2 3/20 0.34
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
F11 P03951 1/20 0.34
TP53 P04637 1/20 0.33
F10 P00742 7/20 0.33
F2 P00734 2/20 0.33
ALDH1A1 P00352 1/20 0.33
PRNP P04156 1/20 0.33
GAA P10253 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5261804 1.00 LEF1 (0.46) LEF1MLLT1MAOAMAOBPYGL
SCHEMBL6838618 0.88 MLLT1 (0.40) MLLT1MAOAMAOBPYGLCTSS
SCHEMBL6838615 0.88 MLLT1 (0.40) MLLT1MAOAMAOBPYGLCTSS
SCHEMBL5255124 0.88 MLLT1 (0.40) MLLT1MAOAMAOBPYGLCTSS
SCHEMBL6839388 0.83 MLLT1 (0.42) MLLT1PYGLCTSSCTSKF10
SCHEMBL5254556 0.83 MLLT1 (0.42) MLLT1PYGLCTSSCTSKF10
SCHEMBL6832182 0.82 MLLT1 (0.36) MLLT1PYGLCTSSCTSKF10
SCHEMBL6832181 0.82 MLLT1 (0.36) MLLT1PYGLCTSSCTSKF10
SCHEMBL6838498 0.82 MLLT1 (0.56) MLLT1PYGLCTSKKDM4ENPC1
SCHEMBL5254519 0.82 MLLT1 (0.56) MLLT1PYGLCTSKKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1453801-B1 SUBSTITUTED 2-AMINO-CYCLOALKANECARBOXAMIDES AND THEIR USE AS CYSTEINE PROTEASE INHIBITORS HOFFMANN LA ROCHE (CH) 2007-03-21 EP disclosed