SCHEMBL5262207

SCHEMBL5262207

CC(CC(=O)O)(NC1=C(c2ccccc2)C(=O)CC1)c1ccc(NC(=O)c2c(Cl)cncc2Cl)cc1

nearest known ligand 0.43

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 20/20 0.43
ITGA4 P13612 20/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6537273 0.83 ITGB1 (0.42) ITGB1ITGA4
SCHEMBL6518083 0.80 ITGB1 (0.49) ITGB1ITGA4
SCHEMBL5260223 0.77 ITGB1 (0.45) ITGB1ITGA4
SCHEMBL5264142 0.74 ITGB1 (0.42) ITGB1ITGA4
SCHEMBL5262203 0.74 ITGB1 (0.43) ITGB1ITGA4
SCHEMBL6514208 0.73 LMNA (0.47) ITGB1ITGA4
SCHEMBL5261193 0.73 ITGB1 (0.42) ITGB1ITGA4
SCHEMBL6512428 0.73 ITGB1 (0.56) ITGB1ITGA4
SCHEMBL5259500 0.72 ITGB1 (0.50) ITGB1ITGA4
SCHEMBL5262425 0.72 ITGB1 (0.44) ITGB1ITGA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1332132-B1 ENAMINE DERIVATIVES AS CELL ADHESION MOLECULES UCB PHARMA SA (BE) 2007-10-10 EP disclosed
US-6780874-B2 AUTOIMMUNE DISEASE; ANTIINFLAMMATORY AGENTS; ANTIPROLIFERATIVE AGENT CELLTECH R & D LIMITED (GB) 2004-08-24 US disclosed
US-6610700-B2 Inhibit binding of integrins to their ligands, use in immune or inflammatory disorders; 3-(4-((2,6-Naphthyridinyl)amino)-phenyl)-2-((2-(1-ethylpropyl)-3-oxo-1 -cyclopentenyl) amino)-propionic acid, for example CELLTECH R & D LIMITED (GB) 2003-08-26 US disclosed