SCHEMBL5262502

SCHEMBL5262502

O=C(O)C1=NCNc2ncccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 3/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
CYP1A2 P05177 2/20 0.39
TNKS2 Q9H2K2 2/20 0.39
KDM4E B2RXH2 4/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
BLM P54132 1/20 0.37
AGER Q15109 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
LMNA P02545 2/20 0.36
P4HTM Q9NXG6 1/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35
KMT2A Q03164 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5220692 0.76 NOS2 (0.53) NAPRTKDM4EL3MBTL1MAPTALDH1A1
Methylamine SCHEMBL27663588 0.72 NOS2 (0.53) SMN1; SMN2KDM4EL3MBTL1MAPTALDH1A1
SCHEMBL3792409 0.71 SMN1; SMN2 (0.40) NAPRTSMN1; SMN2CYP1A2TNKS2KDM4E
SCHEMBL28328220 0.70 NAPRT (0.40) NAPRTSMN1; SMN2CYP1A2KDM4ETDP1
Hydrochloric Acid SCHEMBL5778118 0.70 SMN1; SMN2 (0.39) NAPRTSMN1; SMN2CYP1A2TNKS2KDM4E
SCHEMBL7481174 0.68 CYP1A2 (0.41) SMN1; SMN2CYP1A2TNKS2KDM4ETDP1
SCHEMBL699878 0.66 CYP1A2 (0.58) SMN1; SMN2CYP1A2TNKS2TDP1MAPT
SCHEMBL27456055 0.65 SMN1; SMN2 (0.35) NAPRTSMN1; SMN2CYP1A2TNKS2KDM4E
Methane SCHEMBL7703084 0.64 SMN1; SMN2 (0.34) NAPRTSMN1; SMN2CYP1A2TNKS2KDM4E
SCHEMBL5697942 0.64 CYP1A2 (0.40) SMN1; SMN2CYP1A2TNKS2KDM4ETDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740551-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105760-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed