SCHEMBL5263290

SCHEMBL5263290

O=c1ccc2cnc(Nc3ccc(N4CCC(CCN5CCOCC5)CC4)cc3)nc2n1-c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 15/20 0.67
CCND1 P24385 14/20 0.67
CCND2 P30279 13/20 0.67
CCND3 P30281 13/20 0.67
CDK2 P24941 8/20 0.59
CCNE2 O96020 7/20 0.59
CCNE1 P24864 7/20 0.59
CCNA2 P20248 7/20 0.59
CCNA1 P78396 6/20 0.59
CCNB2 O95067 3/20 0.59
CDK1 P06493 3/20 0.59
CCNB1 P14635 3/20 0.59
CCNB3 Q8WWL7 3/20 0.59
PAK4 O96013 1/20 0.51
PAK1 Q13153 1/20 0.51
PKN1 Q16512 1/20 0.51
JAK3 P52333 4/20 0.51
FGFR1 P11362 4/20 0.51
FGFR2 P21802 4/20 0.51
FGFR4 P22455 4/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5267905 0.88 CDK4 (0.69) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5263285 0.86 CDK4 (0.79) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5269643 0.83 CDK4 (0.49) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5268470 0.83 CDK4 (0.51) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5264126 0.83 CDK4 (0.49) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5267883 0.83 CDK4 (0.75) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5263430 0.83 CDK4 (0.78) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5264503 0.83 CDK4 (0.50) CDK4CCND1CCND2CCND3CDK2
SCHEMBL6807754 0.82 CDK4 (0.48) CDK4CCND1CCND2CCND3CDK2
SCHEMBL5268237 0.81 CDK4 (0.82) CDK4CCND1CCND2CCND3CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1806348-A2 Pyrido (2,3-D)Pyrimidines as inhibitors of cellular proliferation Warner-Lambert Company LLC (US) 2007-07-11 EP disclosed
EP-1255755-A1 PYRIDOPYRIMIDINONE DERIVATIVES FOR TREATMENT OF NEURODEGENERATIVE DISEASE WARNER-LAMBERT COMPANY (US) 2002-11-13 EP disclosed
WO-2001055148-A1 PYRIDOPYRIMIDINONE DERIVATIVES FOR TREATMENT OF NEURODEGENERATIVE DISEASE WARNER-LAMBERT COMPANY (US) 2001-08-02 WO disclosed