SCHEMBL5264073

SCHEMBL5264073

CCOc1cccc(CCNC(=O)c2nc3ccccc3c(=O)[nH]2)c1

nearest known ligand 0.66

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 20/20 0.66
MMP2 P08253 2/20 0.59
MMP10 P09238 2/20 0.59
MMP8 P22894 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4932669 0.91 MMP13 (0.78) MMP13MMP2MMP10MMP8
SCHEMBL4934626 0.90 MMP13 (0.71) MMP13
SCHEMBL689429 0.81 MMP13 (0.80) MMP13MMP2MMP10MMP8
SCHEMBL4934689 0.81 MMP13 (0.84) MMP13
SCHEMBL4936762 0.81 MMP13 (0.67) MMP13MMP2MMP10MMP8
SCHEMBL4934211 0.81 MMP13 (0.84) MMP13
SCHEMBL3641284 0.81 MMP13 (0.86) MMP13
SCHEMBL16562162 0.81 BRD4 (0.61) MMP13
SCHEMBL8279679 0.80 MMP13 (0.73) MMP13MMP2MMP10MMP8
SCHEMBL688369 0.80 MMP13 (1.00) MMP13MMP2MMP10MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740551-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR Takeda Pharmaceutical Company Limited (JP) 2007-01-10 EP disclosed
WO-2005105760-A1 HETEROCYCLIC AMIDE COMPOUND AND USE THEREOF AS AN MMP-13 INHIBITOR TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-10 WO disclosed