SCHEMBL5264441

SCHEMBL5264441

O=C(O)Cc1cnc(-c2ccc(O)cc2)s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.47
CAMK2A Q9UQM7 1/20 0.47
CYP11B1 P15538 1/20 0.47
HSD17B1 P14061 2/20 0.45
HSD17B2 P37059 2/20 0.45
HDAC1 Q13547 4/20 0.40
HDAC2 Q92769 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.40
NAMPT P43490 3/20 0.40
MAPT P10636 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.39
POLB P06746 1/20 0.39
HDAC3 O15379 1/20 0.39
QPCT Q16769 1/20 0.39
NFKB1 P19838 1/20 0.38
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2468247 0.87 ALDH1A1 (0.53) CYP11B1HDAC1HDAC2PTGDR2MAPT
SCHEMBL27682394 0.84 SMN1; SMN2 (0.52) PTGDR2MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL5263509 0.82 PTGDR2 (0.58) CYP11B1HDAC1HDAC2PTGDR2MAPT
SCHEMBL27807801 0.82 MAPT (0.58) HDAC1HDAC2MAPTSMN1; SMN2NPC1
SCHEMBL21229063 0.80 NAMPT (0.45) CYP11B1HSD17B1HSD17B2HDAC1HDAC2
SCHEMBL27717095 0.78 CYP11B1 (0.48) CYP11B1HSD17B1HSD17B2HDAC1HDAC2
SCHEMBL3065978 0.78 CYP11B1 (0.47) CYP11B1HSD17B1HSD17B2HDAC1HDAC2
SCHEMBL27856782 0.78 CSNK2A2 (0.40) CYP11B1HSD17B1HSD17B2HDAC1HDAC2
SCHEMBL4315835 0.77 CYP11B1 (0.65) CYP11B1HSD17B1HSD17B2HDAC1HDAC2
SCHEMBL18641477 0.77 CYP11B1 (0.41) CYP11B1HSD17B1HSD17B2HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1806332-A1 BENZENE COMPOUND HAVING 2 OR MORE SUBSTITUENTS Daiichi Sankyo Company, Limited (JP) 2007-07-11 EP disclosed