SCHEMBL5264577

SCHEMBL5264577

Cc1ccc(N2CCN(C(=O)C3CN(S(=O)(=O)c4ccc(Cl)s4)CC3c3ccccc3)CC2)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.46
MC4R P32245 7/20 0.45
POLB P06746 1/20 0.44
HTT P42858 1/20 0.44
DRD2 P14416 7/20 0.43
DRD4 P21917 5/20 0.43
LMNA P02545 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9926078 1.00 AR (0.46) ARMC4RPOLBHTTDRD2
SCHEMBL9926101 0.93 SMN1; SMN2 (0.47) ARMC4RLMNATSHRMAPK1
SCHEMBL9926090 0.89 AR (0.46) ARMC4RPOLBHTTDRD2
SCHEMBL9926064 0.87 SMN1; SMN2 (0.53) ARMC4RPOLBLMNATSHR
SCHEMBL9926126 0.86 SMN1; SMN2 (0.48) ARMC4RPOLBHTTDRD2
SCHEMBL13987547 0.86 AR (0.46) ARMC4RPOLBHTTDRD2
SCHEMBL5265503 0.86 AR (0.46) ARMC4RPOLBHTTDRD2
SCHEMBL5268950 0.86 MAPT (0.46) ARLMNATSHRMAPK1KMT2A
SCHEMBL9926065 0.86 MAPT (0.46) ARLMNATSHRMAPK1KMT2A
SCHEMBL9925999 0.85 SIGMAR1 (0.53) POLBHTTLMNATSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836180-B1 SULFONYL PYRROLIDINES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS DRUGS SANOFI SA (FR) 2012-06-13 EP disclosed
EP-1836180-A2 SULFONYL PYRROLIDINES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS DRUGS sanofi-aventis (FR) 2007-09-26 EP disclosed
WO-2006072393-A2 SULFONYL PYRROLIDINES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS DRUGS SANOFI-AVENTIS (DE) 2006-07-13 WO disclosed