SCHEMBL5264696

SCHEMBL5264696

Cc1nc(N2CC(CNC(=O)NS(=O)(=O)c3ccccc3)C2)c(C#N)cc1C(=O)O

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 19/20 0.65
RXFP1 Q9HBX9 1/20 0.46
CHRM2 P08172 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
DRD3 P35462 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4105040 0.91 P2RY12 (0.79) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL5592474 0.86 P2RY12 (0.81) P2RY12RXFP1
SCHEMBL5268084 0.85 P2RY12 (0.66) P2RY12CYP3A4CYP2C9
SCHEMBL5264767 0.84 P2RY12 (0.80) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL3922092 0.82 P2RY12 (0.51) P2RY12RXFP1CHRM2CYP3A4CYP2C9
SCHEMBL4565288 0.81 P2RY12 (0.57) P2RY12RXFP1CHRM2CYP3A4CYP2C9
SCHEMBL4105011 0.79 P2RY12 (0.79) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL4109623 0.79 P2RY12 (1.00) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL5592413 0.78 P2RY12 (0.70) P2RY12CHRM2CYP3A4CYP2C9DRD3
SCHEMBL5267177 0.77 P2RY12 (0.69) P2RY12CHRM2CYP3A4CYP2C9DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836189-A1 NOVEL PYRIDINE COMPOUNDS AstraZeneca AB (SE) 2007-09-26 EP disclosed
WO-2006073361-A9 NOVEL PYRIDINE COMPOUNDS ASTRAZENECA AB (SE) 2007-08-02 WO disclosed
WO-2006073361-A1 NOVEL PYRIDINE COMPOUNDS ASTRAZENECA AB (SE) 2006-07-13 WO disclosed